A 67-year-old man with heart failure and atrial fibrillation on digoxin 0.25 mg daily and furosemide presents with nausea, palpitations, and visual halos. Vital signs: BP 128/76 mmHg, HR 102 bpm with irregular rhythm, RR 18, Temp 37°C, SpO2 98%. Serum potassium is 3.0 mEq/L; digoxin level is 2.8 ng/mL (therapeutic: 0.5-2.0). Troponin is normal. Which mechanism explains this drug toxicity?

  1. A)Hypokalemia competitively blocks digoxin cardiac receptors
  2. B)Hypokalemia increases hepatic metabolism of digoxin
  3. C)Hypokalemia increases Na-K-ATPase inhibition by digoxinGABARITO
  4. D)Hypokalemia decreases digoxin protein binding
  5. E)Hypokalemia increases renal clearance of digoxin

Explicação

Digoxin works by inhibiting the Na-K-ATPase pump. Hypokalemia decreases the pump's activity, reducing intracellular potassium. This makes the Na-K-ATPase more susceptible to digoxin inhibition, amplifying digoxin's effects and causing toxicity at therapeutic d... Ver explicação completa e trilha adaptativa →

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